The present invention relates to compounds that are useful as inhibitors
of protein arginine methyltransferase that have a formula selected from
Formula (I), Formula (II) and Formula (III), as well as racemic mixtures,
diastereomers, enantiomers and tautomers thereof and N-oxides, hydrates,
solvates, pharmaceutically acceptable salts, prodrugs and complexes
thereof as defined herein. Said compound are useful as inhibitors of
PRMTs and/or CARM-I. The invention further relates to compositions
comprising such compounds and methods for their use.