Process for preparing water soluble diterpenes and their applications

   
   

Aqueous solutions of diterpenes such as Forskolin, its congeners, analogs and derivatives, up to approximately 6% concentration, are prepared using suitably substituted cyclodextrin as a solubilizing agents. In the absence of cyclodextrin, some diterpenes such as Forskolin are soluble in water only to concentrations of about 0.001%. Such aqueous solutions find applications in topical and systemic use, as pharmaceutical, cosmeceutical, nutraceutical preparations containing diterpenes such as Forskolin and congeners.

De oplossingen in water van diterpenes zoals Forskolin, zijn congeners, analogons en derivaten, tot ongeveer 6% concentratie, worden voorbereid gebruikend geschikt gesubstitueerd cyclodextrien als oplosbaar makende agenten. Bij gebrek aan cyclodextrien, sommige diterpenes zoals Forskolin zijn oplosbaar in water slechts aan concentraties van ongeveer 0.001%. Dergelijke oplossingen in water vinden toepassingen in actueel en systemisch gebruik, zoals farmaceutische, cosmeceutical, nutraceutical voorbereidingen die diterpenes zoals Forskolin en congeners bevatten.

 
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