The present invention relates to 1,3-benzodiazepin-2-ones and 1,3-benzoxazepin-2-ones of formula I: ##STR1## or stereoisomeric forms, stereoisomeric mixtures, or pharmaceutically acceptable salt forms thereof, which are useful as inhibitors of HIV reverse transcriptase, and to pharmaceutical compositions and diagnostic kits comprising the same, and methods of using the same for treating viral infection or as an assay standard or reagent.

A invenção atual relaciona-se a 1,3-benzodiazepin-2-ones e a 1,3-benzoxazepin-2-ones da fórmula I: ## do ## STR1 ou os formulários stereoisomeric, as misturas stereoisomeric, ou pharmaceutically o sal aceitável dão forma disso, que são úteis porque inibidores do transcriptase reverso do HIV, e às composições pharmaceutical e aos jogos diagnósticos que compreendem o mesmo, e aos métodos de usar o mesmo para a infecção viral de tratamento ou que um padrão ou um reagent do assay.

 
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